Pefloxacin mesylate (Standard) (Pefloxacinium mesylate (Standard)) is the analytical standard of Pefloxacin mesylate ( HY-B0147A ). This product is intended for research and analytical applications. Pefloxacin (Pefloxacinium) mesylate is a broad spectrum antibiotic . Pefloxacin blocks DNA replication by inhibiting DNA gyrase . Pefloxacin mesylate inhibits DNA relaxation catalyzed by topoisomerase I with an IC 50 of 45 μg/mL. Pefloxacin mesylate exhibits antibacterial activity against Escherichia coli , Pseudomonas aeruginosa , and Bacteroides fragilis with MIC 90 s of 0.12, 4, and 16 mg/L, respectively. Pefloxacin mesylate has anti- Plasmodium yoelii infection activity. Pefloxacin mesylate increase UVA-induced edema and immunesuppression. Pefloxacin mesylate can be used for infection studies.
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