Pefloxacin (Pefloxacinium) mesylate dihydrate (Standard) is the analytical standard of Pefloxacin mesylate dihydrate ( HY-B0147B ). This product is intended for research and analytical applications. Pefloxacin (Pefloxacinium) mesylate dihydrate is a broad spectrum antibiotic . Pefloxacin mesylate dihydrate blocks DNA replication by inhibiting DNA gyrase . Pefloxacin mesylate dihydrate inhibits DNA relaxation catalyzed by topoisomerase I with an IC 50 of 45 μg/mL. Pefloxacin mesylate dihydrate exhibits antibacterial activity against Escherichia coli , Pseudomonas aeruginosa , and Bacteroides fragilis with MIC 90 s of 0.12, 4, and 16 mg/L, respectively. Pefloxacin mesylate dihydrate has anti- Plasmodium yoelii infection activity. Pefloxacin mesylate dihydrate increase UVA-induced edema and immunesuppression. Pefloxacin mesylate dihydrate can be used for infection studies.
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