Brompheniramine maleate

Overview

Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class. Brompheniramine maleate is a selective histamine H1 receptor antagonist with a K d of 6.06 nM. Brompheniramine maleate can block the hERG channels , calcium channels , and sodium channels with IC 50 s of 0.90 μM, 16.12 μM and 21.26 μM, respectively. Brompheniramine maleate has anticholinergic, antidepressant and anesthetic properties and can be used for allergic rhinitis research.

Application

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Product Information

• Catalog No.: HY-B0480
• CAS No.: 980-71-2
• Molecular Formula: C20H23BrN2O4
• Molecular Weight: 435.31
• Purity: 99.93%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (5.74 mM); Clear solution
• Availability: In-stock

Source

Original product source