Brompheniramine

Overview

Brompheniramine ((±)-Brompheniramine) is a potent and orally active antihistamine of the alkylamine class. Brompheniramine is a selective histamine H1 receptor antagonist with a K d of 6.06 nM. Brompheniramine can block the hERG channels , calcium channels , and sodium channels with IC 50 s of 0.90 μM, 16.12 μM and 21.26 μM, respectively. Brompheniramine has anticholinergic, antidepressant and anesthetic properties and can be used for allergic rhinitis research.

Application

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Product Information

• Catalog No.: HY-B0480A
• CAS No.: 86-22-6
• Molecular Formula: C16H19BrN2
• Molecular Weight: 319.24
• Purity: 99.82%
• Storage: Pure form -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source