AZ-5104

Overview

AZ-5104 is an active, demethylated metabolite of AZD 9291. AZ-5104 is an EGFR inhibitor with IC 50 s of 1, 6, 1, 25 and 7 nM for EGFR L858R/T790M , EGFR L858R , EGFR L861Q , EGFR and ErbB4, respectively.

Application

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Product Information

• Catalog No.: HY-B0793
• CAS No.: 1421373-98-9
• Molecular Formula: C27H31N7O2
• Molecular Weight: 485.58
• Purity: 99.91%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (5.15 mM); Clear solution
• Availability: In-stock

Source

Original product source