WAY 208466 dihydrochloride is a potent and selective 5-HT 6 receptor agonist ( EC 50 =7.3 nM for the human 5-HT 6 receptor). WAY-208466 dihydrochloride elevates cortical GABA levels in rat frontal cortex. WAY 208466 dihydrochloride exhibits antidepressant and anxiolytic-like effects.
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