Azepexole dihydrochloride

Overview

Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pK i s of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC 50 = 78.72 nM).

Application

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Product Information

• Catalog No.: HY-103212
• CAS No.: 36067-72-8
• Molecular Formula: C9H17Cl2N3O
• Molecular Weight: 254.16
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source