Chlorphenoxamine, an antihistamine and anticholinergic agent is a GPCR antagonist. Chlorphenoxamine inhibits multiple lethal viral diseases, such as SARS-CoV , MERS-CoV , EBOV and malaria . Chlorphenoxamine shows anti-filovirus activity against both EBOV and Marburg virus ( MARV ) with IC 50 s of 1.1 μM and 6.2 μM, respectively. Chlorphenoxamine is used for allergic conditions, urticaria, viral diseases and Parkinson’s disease.
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