Tracazolate hydrochloride

Overview

Tracazolate (ICI 136753) hydrochloride is a potent GABA A receptor modulator. Tracazolate hydrochloride has selectivity for β3 and potentiates α1β1γ2s (EC 50 =13.2 μM), α1β3γ2 (EC 50 =1.5 μM). Tracazolate hydrochloride has the potency (EC 50 ) determined by the nature of the third subunit (γ1-3, δ, ε) within the receptor complex. Tracazolate hydrochloride possesses anxiolytic and anticonvulsant activity.

Application

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Product Information

• Catalog No.: HY-B1803A
• CAS No.: 1135210-68-2
• Molecular Formula: C16H25ClN4O2
• Molecular Weight: 340.85
• Purity: 99.24%
• Storage: -20°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Availability: In-stock

Source

Original product source