Melperone (Standard)

Overview

Melperone (Standard) is the analytical standard of Melperone ( HY-B2169 ). This product is intended for research and analytical applications. Melperone is a butyrophenone with atypical antipsychotic properties. Melperone is a multireceptor antagonist with K d s of 102 nM, 180 nM, 180 nM, and 150 nM for 5-HT2A , dopamine D2 , α1-adrenergic , and α2-adrenergic receptors , respectively. Melperone has weak binding to histamine H1, 5-HT2C, 5-HT1A, 5-HT1D, and muscarinic receptors, with K d values ​​of 580 nM, 2100 nM, 2200 nM, 3400 nM, >10000 nM, respectively. Melperone is also a CYP2D6 inhibitor. Melperone can be used for the study of schizophrenia, and agitation in the elderly.

Application

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Product Information

• Catalog No.: HY-B2169R
• CAS No.: 3575-80-2
• Molecular Formula: C16H22FNO
• Molecular Weight: 263.35
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source