Melperone-d 4 hydrochloride

Overview

Melperone-d 4 hydrochloride is the deuterium labeled Melperone hydrochloride ( HY-103109 ). Melperone hydrochloride is a butyrophenone with atypical antipsychotic properties. Melperone hydrochloride is a multireceptor antagonist with K d s of 102 nM, 180 nM, 180 nM, and 150 nM for 5-HT2A , dopamine D2 , α1-adrenergic , and α2-adrenergic receptors , respectively. Melperone hydrochloride has weak binding to histamine H1, 5-HT2C, 5-HT1A, 5-HT1D, and muscarinic receptors, with K d values ​​of 580 nM, 2100 nM, 2200 nM, 3400 nM, >10000 nM, respectively. Melperone hydrochloride is also a CYP2D6 inhibitor. Melperone hydrochloride can be used for the study of schizophrenia, and agitation in the elderly.

Application

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Product Information

• Catalog No.: HY-B2169S2
• CAS No.: 1219798-80-7
• Molecular Formula: C16H19D4ClFNO
• Molecular Weight: 303.84
• Purity: 99.84%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Availability: In-stock

Source

Original product source