Pinoresinol Diglucoside is an orally active lignan with multifunctional bioactivity. Pinoresinol Diglucoside interacts with targets including ALB , HIF1A , GSK3B , BCL2 , MARK3 , IL6 , NF-κB p65 , Nrf2 , HO-1 , and TLR4 , and modulates pathways including PI3K-Akt , estrogen, MAPK , Rap1 , AKT/mTOR/NF-κB , and TGF-β1/Smads . Pinoresinol Diglucoside regulates osteogenesis, bone resorption, oxidative stress, inflammation, apoptosis , ferroptosis , ferritinophagy, cardiac fibrosis, and vasorelaxation. Pinoresinol Diglucoside can be used for the research of osteoporosis, ischemia/reperfusion-induced brain injury, Alzheimer’s disease, myocardial ischemia-reperfusion injury, chondrodysplasia, diabetic cardiomyopathy, cardiac hypertrophy, hypertension, cisplatin-induced hearing loss, atherosclerotic cardiovascular diseases, and disuse osteoporosis.
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