Cabotegravir (GSK744, GSK1265744)

Overview

Cabotegravir (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor against a broad range of HIV subtypes, and inhibits the HIV-1 integrase catalyzed strand transfer reaction with IC50 of 3.0 nM. Phase 2.

Application

Products > Drug Discovery > Inhibitor | Products > Drug Discovery > Inhibitor | Infection | HIV Integrase

Product Information

• Catalog No.: B0084-463362
• CAS No.: 1051375-10-0
• Molecular Formula: C19H17F2N3O5
• Molecular Weight: 405.35
• Purity: >98%
• Storage: Store at -20°C
• Solubility: In Vitro : DMSO : 16.67 mg/mL(41.12 mM;Need ultrasonic) In Vivo: 1.Add each solvent one by one:10% DMSO >> 90%corn oil Solubility: ≥ 1.67 mg/mL (4.12 mM); Clear solution

Source

Original product source