PF 04531083

Overview

PF 04531083 is an orally active and selective Na V 1.8 blocker with an IC 50 of 0.7 μM. PF 04531083 is a blood-brain barrier (BBB) penetrant compound. PF 04531083 can be used for the research of respiratory system and neuropathic/inflammatory pain.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Sodium Channel

Product Information

• Catalog No.: HY-105283
• CAS No.: 1079400-07-9
• Molecular Formula: C17H16ClN5O2
• Molecular Weight: 357.79
• Purity: 99.62%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.08 mg/mL (5.81 mM); Clear solution
• Availability: In-stock

Source

Original product source