Miltirone is an orally active natural compound found in the root of Salvia miltiorrhiza. Miltirone is a central benzodiazepine receptor partial agonist, with an IC50 of 0.3 μM. Miltirone induces ROS - and-p53 dependent apoptosis . Miltirone inhibits carboxylesterase 2 ( CES2 ; Ki = 0.04 μM) and SARS-CoV main protease (Mpro).
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