Sarpogrelate hydrochloride

Overview

Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT 2 R antagonist, with pK i s of 8.52, 6.57, and 7.43 for 5-HT 2A , 5-HT 2B , and 5-HT 2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT 1 , 5-HT 3 , 5-HT 4 , α 1 -, α 2 - and β-adrenoreceptor, histamine H 1 , H 2 and muscarinic M 3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis.

Application

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Product Information

• Catalog No.: HY-10564
• CAS No.: 135159-51-2
• Molecular Formula: C24H32ClNO6
• Molecular Weight: 465.97
• Purity: 99.09%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (5.37 mM); Clear solution
• Availability: In-stock

Source

Original product source