Lurosetron

Overview

Lurosetron (GR-87442) is a 6-fluoro analogue of Alosetron ( HY-70050A ). Lurosetron is a serotonin 5-HT3 receptor antagonist. Lurosetron inhibits recombinant (rbt) CYP1A2 , with an IC 50 of 0.1 μM. Lurosetron also inhibits other CYP isoforms, including rbtCYP2C9 and rbtCYP3A4 with IC 50 s ranging between 3.5 μM and 16 μM..

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > 5-HT Receptor

Product Information

• Catalog No.: HY-106379
• CAS No.: 128486-54-4
• Molecular Formula: C17H17FN4O
• Molecular Weight: 312.34
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source