CBP-1018 is a PDC (peptide-drug conjugate) formed by conjugating Monomethyl auristatin E ( HY-15162 ) to a dual-targeting ligand of FLOR1 / PSMA (prostate-specific membrane antigen) via a linker ( HY-78738 ). CBP-1018 binds to FLOR1 and prostate-specific membrane antigen ( PSMA ). CBP-1018 is applicable to the research of solid tumors and metastatic castration-resistant prostate cancer .
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