Cyclic(YCDGFYACYMDV)

Cyclic(YCDGFYACYMDV)
  • CAS No.:535959-77-4
  • Grade:99.98%
  • Formula:C65H82N12O20S3
  • M.W.:1447.61

Overview

Cyclic(YCDGFYACYMDV) is a HER2 signaling pathway inhibitor with anti-cancer activity. This compound self-assembles into nanoparticles in aqueous solution and transforms into nanofibers upon specific binding to HER2 on cancer cells. This transformation disrupts HER2 dimerization and subsequent downstream signaling events, leading to cancer cell apoptosis ( Apoptosis ). The inhibitory effects on HER2 positive breast cancer have been demonstrated to be effective in a murine xenograft model.

Application

Products | Products > Peptides | Products > Signaling Pathways > JAK/STAT Signaling | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Signaling Pathways > Apoptosis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > EGFR | Products > Signaling Pathways > Apoptosis

Product Information

  • Catalog No.: HY-P10793
  • CAS No.: 535959-77-4
  • Molecular Formula: C65H82N12O20S3
  • Molecular Weight: 1447.61
  • Purity: 99.98%
  • Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source


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