Octoclothepin maleate salt

Overview

Octoclothepin (Clorotepine) maleate salt is a D 2 dopamine receptor antagonist and 5-HT 2 serotonin receptor antagonist , with K i values of 0.67 nM, 0.57 nM, and 0.19 nM for the dopamine D 2 , 5-HT 2A , and 5-HT 2C receptors, respectively. Octoclothepin maleate salt also binds to adrenergic receptors , with K i values of 0.66 nM, 0.56 nM, and 0.77 nM for α 1a , α 1b , and α 1d , respectively. Octoclothepin maleate salt can be used in schizophrenia research.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > Others | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Drug Derivative | Products > Signaling Pathways > 5-HT Receptor

Product Information

• Catalog No.: HY-106587A
• CAS No.: 4789-68-8
• Molecular Formula: C23H25ClN2O4S
• Molecular Weight: 460.97
• Purity: 98.81%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.5 mg/mL (5.42 mM); Clear solution
• Availability: In-stock

Source

Original product source