Anrikefon

Overview

Anrikefon is a peripherally restricted kappa opioid receptor (KOR) agonist, with an IC 50 of 0.54 nM, an EC 50 of 2.41 pM, and a K a of 0.068 nM against human KOR , and it exhibits high selectivity over μ and δ opioid receptors. Anrikefon exerts analgesic effects by inhibiting behaviors associated with inflammatory, postoperative and neuropathic pain, and also exerts antipruritic effects by reducing itch-related behaviors. Anrikefon can be used in research on pain, pruritus, and pruritus associated with chronic kidney disease.

Application

Products | Products > Peptides | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Opioid Receptor

Product Information

• Catalog No.: HY-P3445
• CAS No.: 2269511-95-5
• Molecular Formula: C39H57N7O5
• Molecular Weight: 703.91
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source