MK-0249

Overview

MK-0249 (Compound 1) is a potent, selective and orally active histamine H 3 receptor antagonist, with an IC 50 of 1.7 nM for human H3.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > Immunology/Inflammation | Products > Research Areas > Neurological Disease | Products > Research Areas > Endocrinology | Products > Signaling Pathways > Histamine Receptor

Product Information

• Catalog No.: HY-U00076
• CAS No.: 862309-06-6
• Molecular Formula: C23H24F3N3O2
• Molecular Weight: 431.45
• Purity: 98.28%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 1.25 mg/mL (2.90 mM); Clear solution
• Availability: In-stock

Source

Original product source