2-Aminoethyl diphenylborinate

Overview

2-Aminoethyl diphenylborinate (2-APB) is a cell-permeable inhibitor of Inositol triphosphate receptor ( IP3R ). 2-Aminoethyl diphenylborinate also inhibits the store-operated Ca 2+ (SOC) channel and activates some TRP channels (V1, V2 and V3). Additionally, 2-Aminoethyl diphenylborinate has inhibitory effects on vasospasm. At high concentrations, it exhibits specific anti-inflammatory and antioxidant effects in neural tissue.

Application

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Product Information

• Catalog No.: HY-W009724
• CAS No.: 524-95-8
• Molecular Formula: C14H16BNO
• Molecular Weight: 225.09
• Purity: 98.86%
• Storage: Powder -20°C, 3 years , 4°C, 2 years * The compound is unstable in solutions, freshly prepared is recommended.
• Solubility: ≥ 2.08 mg/mL (9.24 mM); Clear solution
• Availability: In-stock

Source

Original product source