PT2399

Overview

PT2399 is a potent and selective HIF-2α antagonist, which directly binds to HIF-2α PAS B domain with an IC 50 of 6 nM. PT2399 displays potent antitumor activity in vivo.

Application

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Product Information

• Catalog No.: HY-108697
• CAS No.: 1672662-14-4
• Molecular Formula: C17H10F5NO4S
• Molecular Weight: 419.32
• Purity: 99.96%
• Storage: -20°C, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
• Solubility: ≥ 1.67 mg/mL (3.98 mM); Clear solution
• Availability: In-stock

Source

Original product source