Abexinostat (CRA 024781) is a novel pan- HDAC inhibitor mostly targeting HDAC1 with K i of 7 nM. Abexinostat also inhibits metallo-β-lactamase domain-containing protein 2 ( MBLAC2 ) hydrolase activity with an EC 50 below 10 nM.
Products | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > HDAC
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