CGP60474

Overview

CGP60474, a highly potent anti-endotoxemic agent, is a potent cyclin-dependent kinase ( CDK ) inhibitor ( IC 50 values are 26, 3, 4, 216, 10, 200 and 13 nM for CDK1/B, CDK2/E, CDK2/A, CDK4/D, CDK5/p25, CDK7/H and CDK9/T, respectively). CGP60474 is a selective and ATP-competitive PKC inhibitor.

Application

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Product Information

• Catalog No.: HY-11009
• CAS No.: 164658-13-3
• Molecular Formula: C18H18ClN5O
• Molecular Weight: 355.82
• Purity: 98.90%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (7.03 mM); Clear solution
• Availability: In-stock

Source

Original product source