PPARα/δ antagonist-1

Overview

PPARα/δ antagonist-1 is an orally active, highly selective dual antagonist of PPARα/δ , with IC 50 values of 0.113 μM and 0.025 μM against human PPARα and PPARδ , respectively. PPARα/δ antagonist-1 exhibits an excellent in vitro activity profile and preliminary efficacy in mouse tumor models. PPARα/δ antagonist-1 can be used in studies related to cancers (melanoma metastasis, ovarian cancer ).

Application

Products | Products > Disease Areas > Urogenital Cancer | Products > Disease Areas > Metastatic Melanoma | Products > Disease Areas > Cancer | Products > Disease Areas > Urogenital Disease | Products > Disease Areas > Melanoma | Products > Disease Areas > Ovarian Cancer | Products > Signaling Pathways > Cell Cycle/DNA Damage | Products > Signaling Pathways > Vitamin D Related/Nuclear Receptor | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > PPAR

Product Information

• Catalog No.: HY-182619
• CAS No.: 1673590-38-9
• Molecular Formula: C34H29F4N3O4
• Molecular Weight: 619.61
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source