Tizaterkib

Tizaterkib
  • CAS No.:2097416-76-5
  • Grade:99.10%
  • Formula:C24H24F2N8O2
  • M.W.:494.50
  • Solvent:≥ 2.08 mg/mL (4.21 mM); Clear solution

Overview

Tizaterkib (AZD0364) is a potent and selective ERK2 inhibitor extracted from patent WO2017080979A1, compound example 18, has an IC 50 of 0.6 nM.

Application

Products | Products > Signaling Pathways > MAPK/ERK Pathway | Products > Signaling Pathways > Stem Cell/Wnt | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Stem Cells | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > ERK

Product Information

  • Catalog No.: HY-111483
  • CAS No.: 2097416-76-5
  • Molecular Formula: C24H24F2N8O2
  • Molecular Weight: 494.50
  • Purity: 99.10%
  • Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
  • Solubility: ≥ 2.08 mg/mL (4.21 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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