Bobcat339

Overview

Bobcat339 is a potent and selective cytosine-based inhibitor of TET enzyme , with IC 50 s of 33 μM and 73 μM for TET1 and TET2 , respectively. Bobcat339 is useful to the field of epigenetics and serves as a starting point for new therapeutics that target DNA methylation and gene transcription.

Application

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Product Information

• Catalog No.: HY-111558
• CAS No.: 2280037-51-4
• Molecular Formula: C16H12ClN3O
• Molecular Weight: 297.74
• Purity: 99.44%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: 2.5 mg/mL (8.40 mM); Clear solution; Need ultrasonic
• Availability: In-stock

Source

Original product source