GS-626510

Overview

GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with K d values of 0.59-3.2 nM for BRD2/3/4, with IC 50 values of 83 nM and 78 nM foe BD1 and BD2, respectively.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Epigenetic Reader Domain

Product Information

• Catalog No.: HY-114416
• CAS No.: 1637770-13-8
• Molecular Formula: C25H22N4O
• Molecular Weight: 394.47
• Purity: 99.46%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (6.34 mM); Clear solution
• Availability: In-stock

Source

Original product source