GSK467

Overview

GSK467 is a cell penetrant and selective KDM5B (JARID1B or PLU1) inhibitor with a K i of 10 nM and an IC 50 of 26 nM. GSK467 shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members.

Application

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Product Information

• Catalog No.: HY-116761
• CAS No.: 1628332-52-4
• Molecular Formula: C17H13N5O2
• Molecular Weight: 319.32
• Purity: 99.34%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: 2.08 mg/mL (6.51 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source