MRS 1523

Overview

MRS 1523 is a potent and selective adenosine A 3 receptor antagonist with K i values of 18.9 nM and 113 nM for human and rat A 3 receptors , respectively. In rat this corresponds to selectivities of 140- and 18-fold vs A 1 and A 2A receptors, respectively. MRS 1523 can exert antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons.

Application

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Product Information

• Catalog No.: HY-121119
• CAS No.: 212329-37-8
• Molecular Formula: C23H29NO3S
• Molecular Weight: 399.55
• Purity: 99.97%
• Storage: Pure form -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (6.26 mM); Clear solution
• Availability: In-stock

Source

Original product source