AKR1C2/3-IN-2

Overview

AKR1C2/3-IN-2 is a potential AKR1C3 inhibitor with selective AKR1C3 activity. AKR1C2/3-IN-2 is able to block AKR1C3-mediated testosterone (T) production and PSA induction, affecting the endocrine activity of prostate cancer cells. AKR1C2/3-IN-2 shows selectivity over other AKR1C enzymes , indicating its potential application in inhibiting drug-resistant prostate cancer . AKR1C2/3-IN-2 has no inhibitory activity against COX isomerases, further emphasizing its specificity as a prostate cancer inhibitory compound.

Application

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Product Information

• Catalog No.: HY-121656
• CAS No.: 56600-73-8
• Molecular Formula: C15H16O3
• Molecular Weight: 244.29
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source