TG2 inhibitor VA4

Overview

TG2 inhibitor VA4 (compound VA4) is an irreversible Type 2 transglutaminase (TG2) inhibitor. TG2 inhibitor VA4 reacts exclusively at the TG2 transamidase site, inhibits both transamidase and GTP-binding activities.

Application

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Product Information

• Catalog No.: HY-122709
• CAS No.: 2088001-23-2
• Molecular Formula: C33H41N5O6S
• Molecular Weight: 635.77
• Purity: 99.66%
• Storage: 4°C, sealed storage, away from moisture and light * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
• Solubility: ≥ 2.5 mg/mL (3.93 mM); Clear solution
• Availability: In-stock

Source

Original product source