Borussertib

Overview

Borussertib, a chemical probe, is a covalent-allosteric and first-in-class inhibitor of protein kinase Akt , with an IC 50 of 0.8 nM and a K i of 2.2 nM for Akt wt .

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PI3K/Akt/mTOR | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Immunotherapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Akt

Product Information

• Catalog No.: HY-122913
• CAS No.: 1800070-77-2
• Molecular Formula: C36H32N6O3
• Molecular Weight: 596.68
• Purity: 99.18%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.08 mg/mL (3.49 mM); Clear solution
• Availability: In-stock

Source

Original product source