BI-2545

Overview

BI-2545, a chemical probe, is a potent autotaxin (ATX) inhibitor that significantly reduces LPA, with IC 50 s of 2.2 nM and 3.4 nM for human ATX and rat ATX, respectively.

Application

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Product Information

• Catalog No.: HY-124772
• CAS No.: 2162961-71-7
• Molecular Formula: C23H19F6N5O3
• Molecular Weight: 527.42
• Purity: 98.85%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.08 mg/mL (3.94 mM); Clear solution
• Availability: In-stock

Source

Original product source