ZEN-2759

Overview

ZEN-2759 is a potent BET (Bromodomain and Extra-Terminal Domain) inhibitor, with IC 50 values of 0.23, 0.08 and 0.28 μM for BRD4(BD1) , BRD4(BD2) , and BRD4(BD1BD2) , respectively.

Application

Products | Products > Disease Areas > Cancer | Products > Disease Areas > Blood or Cardio-cerebrovascular Disease | Products > Disease Areas > Leukemia/Lymphoma/Myeloma | Products > Disease Areas > Blood Disease | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > Epigenetic Reader Domain

Product Information

• Catalog No.: HY-129201
• CAS No.: 1616400-50-0
• Molecular Formula: C17H16N2O2
• Molecular Weight: 280.32
• Purity: 99.51%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (8.92 mM); Clear solution
• Availability: In-stock

Source

Original product source