(S)-PI3Kα-IN-4

Overview

(S)-PI3Kα-IN-4 is a potent inhibitor of PI3Kα , with an IC 50 of 2.3 nM. (S)-PI3Kα-IN-4 shows 38.3-, 4.25-, and 4.93-fold selectivity for PI3Kα over PI3Kβ , PI3Kδ , and PI3Kγ , respectively. (S)-PI3Kα-IN-4 can be used for the research of cancer .

Application

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Product Information

• Catalog No.: HY-131345A
• CAS No.: 2322293-84-3
• Molecular Formula: C25H23ClFN5O5S
• Molecular Weight: 560.00
• Purity: 99.77%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (4.46 mM); Clear solution
• Availability: In-stock

Source

Original product source