I-BET151

Overview

I-BET151 (GSK1210151A) is a BET bromodomain inhibitor which inhibits BRD4 , BRD2 , and BRD3 with pIC 50 of 6.1, 6.3, and 6.6, respectively.

Application

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Product Information

• Catalog No.: HY-13235
• CAS No.: 1300031-49-5
• Molecular Formula: C23H21N5O3
• Molecular Weight: 415.44
• Purity: 99.47%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (6.02 mM); Clear solution
• Availability: In-stock

Source

Original product source