(s)-PF-4136309

Overview

(s)-PF-4136309 is the isomer of PF-4136309 ( HY-13245 ), and can be used as an experimental control. PF-4136309 is a potent, selective, and orally bioavailable CCR2 antagonist, with IC 50 s of 5.2 nM, 17 nM and 13 nM for human, mouse and rat CCR2 .

Application

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Product Information

• Catalog No.: HY-13245A
• CAS No.: 1372407-07-2
• Molecular Formula: C29H31F3N6O3
• Molecular Weight: 568.59
• Purity: 98.93%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source