PKCβ inhibitor 1

Overview

PKCβ inhibitor 1 is a potent, ATP-competitive, and selective PKCβ inhibitor with IC 50 s of 21 and 5 nM for human PKCβ1 and PKCβ2, respectively. PKCβ inhibitor 1 exhibits selectivity of more than 60-fold in favor of PKCβ2 relative to other PKC isozymes ( PKCα , PKCγ , and PKCε ).

Application

Products | Products > Signaling Pathways > Epigenetics | Products > Signaling Pathways > TGF-beta/Smad | Products > Signaling Pathways > Apoptosis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > PKC | Products > Signaling Pathways > Apoptosis

Product Information

• Catalog No.: HY-13335
• CAS No.: 257879-35-9
• Molecular Formula: C24H21N5O2
• Molecular Weight: 411.46
• Purity: 99.40%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 6.25 mg/mL (15.19 mM); Clear solution
• Availability: In-stock

Source

Original product source