PF-8380

Overview

PF-8380 is a potent autotaxin inhibitor with an IC 50 of 2.8 nM in isolated enzyme assay and 101 nM in human whole blood.

Application

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Product Information

• Catalog No.: HY-13344
• CAS No.: 1144035-53-9
• Molecular Formula: C22H21Cl2N3O5
• Molecular Weight: 478.33
• Purity: 99.05%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 0.67 mg/mL (1.40 mM); Clear solution
• Availability: In-stock

Source

Original product source