EN4

Overview

EN4 is a covalent ligand that targets cysteine 171 (C171) of MYC . EN4 is selective for c-MYC over N-MYC and L-MYC. EN4 inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis.

Application

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Product Information

• Catalog No.: HY-134761
• CAS No.: 1197824-15-9
• Molecular Formula: C25H24N2O4
• Molecular Weight: 416.47
• Purity: 96.29%
• Storage: 4°C, protect from light * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
• Solubility: 2.08 mg/mL (4.99 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source