(R,R)-CPI-1612

Overview

(R,R)-CPI-1612 is the isomer of CPI-1612 ( HY-136285 ), and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC 50 of 8.1 nM for EP300 HAT . CPI-1612 has an anticancer activity.

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Epigenetics | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Histone Acetyltransferase

Product Information

• Catalog No.: HY-136285A
• CAS No.: 2374972-35-5
• Molecular Formula: C27H26N6O
• Molecular Weight: 450.53
• Purity: 99.49%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 3.25 mg/mL (7.21 mM); Clear solution
• Availability: In-stock

Source

Original product source