BC-DXI-843

BC-DXI-843
  • CAS No.:2421117-98-6
  • Grade:99.76%
  • Formula:C28H26N4O4S2
  • M.W.:546.66
  • Solvent:≥ 2.08 mg/mL (3.80 mM); Clear solution

Overview

BC-DXI-843 is a potent and specific AIMP2-DX2 inhibitor with an IC 50 of 0.92 μM, more than 100-fold selectivity over AIMP2 (IC 50 >100 μM) in a luciferase assay. BC-DXI-843 acts as a promising lead targeting AIMP2-DX2 in lung cancer .

Application

Products | Products > Disease Areas > Cancer | Products > Disease Areas > Lung Cancer | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Signaling Pathways > Aminoacyl-tRNA Synthetase

Product Information

  • Catalog No.: HY-136431
  • CAS No.: 2421117-98-6
  • Molecular Formula: C28H26N4O4S2
  • Molecular Weight: 546.66
  • Purity: 99.76%
  • Storage: 4°C, protect from light * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
  • Solubility: ≥ 2.08 mg/mL (3.80 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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