SAR502250

Overview

SAR502250 is a potent, selective, ATP competitive, orally active and brain-penetrant inhibitor of GSK3 , with an IC 50 of 12 nM for human GSK-3β . SAR502250 displays antidepressant-like activity. SAR502250 can be used for the research of Alzheimer’s disease (AD).

Application

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Product Information

• Catalog No.: HY-137472
• CAS No.: 503860-57-9
• Molecular Formula: C19H18FN5O2
• Molecular Weight: 367.38
• Purity: 99.29%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (6.80 mM); Clear solution
• Availability: In-stock

Source

Original product source