JANEX-1 (WHI-P131) hydrochloride is a potent and specific JAK3 inhibitor ( K i =2.3 μM). JANEX-1 hydrochloride shows potent JAK3 inhibitory activity ( IC 50 =78 μM), does not inhibit JAK1 and JAK2 .
Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > Epigenetics | Products > Signaling Pathways > Stem Cell/Wnt | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Signaling Pathways > JAK/STAT Signaling | Products > Research Areas > Cancer > Cancer Stem Cells | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > JAK
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