(R)-PS210

Overview

(R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC 50 value of 1.8 μM. (R)-PS210 targets to the PIF-binding pocket of?PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-interacting fragment.

Application

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Product Information

• Catalog No.: HY-13856
• CAS No.: 1410101-89-1
• Molecular Formula: C19H15F3O5
• Molecular Weight: 380.31
• Purity: 98.09%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 5.75 mg/mL (15.12 mM); Clear solution
• Availability: In-stock

Source

Original product source