Bisindolylmaleimide I hydrochloride

Overview

Bisindolylmaleimide I (GF109203X) hydrochloride is a cell-permeable and reversible PKC inhibitor ( IC 50 of 20 nM, 17 nM, 16 nM, and 20 nM for PKCα , PKCβI, PKCβII, and PKCγ . Bisindolylmaleimide I hydrochloride is also a GSK-3 inhibitor.

Application

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Product Information

• Catalog No.: HY-13867A
• CAS No.: 176504-36-2
• Molecular Formula: C25H25ClN4O2
• Molecular Weight: 448.94
• Purity: 98.44%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: 2.08 mg/mL (4.63 mM); Suspended solution; Need ultrasonic
• Availability: In-stock

Source

Original product source