N-Desethyl Sunitinib hydrochloride

Overview

N-Desethyl Sunitinib (SU-12662) (hydrochloride) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR , PDGFRβ and KIT inhibitor with K i values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively.

Application

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Product Information

• Catalog No.: HY-138813
• CAS No.: 1261432-05-6
• Molecular Formula: C20H24ClFN4O2
• Molecular Weight: 406.88
• Purity: 99.14%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: 2.5 mg/mL (6.14 mM); Clear solution; Need ultrasonic
• Availability: In-stock

Source

Original product source